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Chemical compound
Relugolix, sold under the brand names Orgovyx and Relumina among others, is a gonadotropin-releasing hormone antagonist (GnRH receptor antagonist) medication
Relugolix
Combination medication
Relugolix/estradiol/norethisterone acetate, sold under the brand names Myfembree and Ryeqo, is a fixed-dose combination hormonal medication which is used
Relugolix/estradiol/norethisterone acetate
Relugolix/estradiol/norethisterone_acetate
Class of medications
antagonistic effect, while other GnRH antagonists, such as elagolix and relugolix, are non-peptide and small-molecule compounds. GnRH antagonists compete
Gonadotropin-releasing hormone antagonist
Gonadotropin-releasing_hormone_antagonist
Gonadotropin secreted by the adenohypophysis
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Luteinizing_hormone
Chemical compound
introduction of elagolix in the United States and Canada was followed by that of relugolix (brand name Relumina), the next second-generation GnRH antagonist, in
Elagolix
Type of medication which modulates the GnRH receptor
are structurally related to GnRH – or small-molecules like elagolix and relugolix, which are structurally distinct from and unrelated to GnRH analogues
Gonadotropin-releasing hormone modulator
Gonadotropin-releasing_hormone_modulator
Male reproductive organ cancer
symptoms of metastases. In these people, GnRH antagonists like degarelix or relugolix are given instead, and can also rapidly reduce testosterone levels. Reducing
Prostate_cancer
Chemical compound
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Buserelin
Manufactured (artificial) injectable hormone
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Leuprorelin
Drug class affecting sex hormones
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Gonadotropin-releasing hormone agonist
Gonadotropin-releasing_hormone_agonist
Medication used to inhibit puberty
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Puberty_blocker
Hormone for the maternal recognition of pregnancy
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Human_chorionic_gonadotropin
Gender-affirming medical treatment
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Gender-affirming hormone therapy
Gender-affirming_hormone_therapy
Gonadotropin that regulates the development of reproductive processes
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Follicle-stimulating_hormone
Drug class
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Progonadotropin
Pharmaceutical drug
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Menotropin
Type of medication
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Gonadotropin_preparations
Glycoprotein polypeptide hormones
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Gonadotropin
Type of gender-affirming medical treatment
non-peptide and orally active GnRH antagonists, elagolix (Orilissa) and relugolix (Relumina), were introduced for medical use in 2018 and 2019, respectively
Feminizing_hormone_therapy
Pharmaceutical drug
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Ganirelix
Class of pharmaceutical drugs
orally active GnRH antagonist to be introduced for medical use 2019: Relugolix is the second orally active GnRH antagonist to be introduced for medical
Antiandrogen
GnRH-agonist
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Triptorelin
Chemical compound
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Gonadorelin
Chemical compound
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Goserelin
G-protein coupled receptor
Cetrorelix Degarelix Ganirelix Ozarelix Elagolix Linzagolix Opigolix Relugolix Sufugolix Current research is looking into pharmacoperones, or chemical
Gonadotropin-releasing hormone receptor
Gonadotropin-releasing_hormone_receptor
Chemical compound
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Degarelix
Drug used in IVF procedures
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Cetrorelix
Drug
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Antigonadotropin
Mammalian protein found in Homo sapiens
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Gonadotropin-releasing hormone
Gonadotropin-releasing_hormone
Transmembrane receptor found in humans
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Luteinizing hormone/choriogonadotropin receptor
Luteinizing_hormone/choriogonadotropin_receptor
Pharmaceutical compound
Teverelix (antarelix); Non-peptides: Elagolix Linzagolix Merigolix Opigolix Relugolix Sufugolix Gonadotropin LH/hCGTooltip Luteinizing hormone/choriogonadotropin
Merigolix
Chemical compound
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Opigolix
years. The National Institute of Health and Care Excellence approves relugolix, used to treat the symptoms of endometriosis, for use by the NHS in England
2025_in_the_United_Kingdom
Pharmaceutical drug classification
H01CC04 Linzagolix H01CC53 Elagolix, estradiol and norethisterone H01CC54 Relugolix, estradiol and norethisterone "ATC (Anatomical Therapeutic Chemical Classification
ATC_code_H01
Type of gender-affirming medical treatment
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Masculinizing_hormone_therapy
Pharmaceutical drug classification
Exemestane L02BX01 Abarelix L02BX02 Degarelix L02BX03 Abiraterone L02BX04 Relugolix L02BX53 Abiraterone and corticosteroids "ATC (Anatomical Therapeutic Chemical
ATC_code_L02
Chemical compound
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Linzagolix
Pharmaceutical drug
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Nafarelin
Chemical compound
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Deslorelin
Chemical compound
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Histrelin
Pharmaceutical drug classification
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
ATC_code_G
Investigational PMS/PMDD drugs
GnRH agonists (e.g., leuprorelin) and GnRH antagonists (e.g., elagolix, relugolix) (with or without add-back estrogen–progestogen therapy) Neurosteroids
List of investigational PMS/PMDD drugs
List_of_investigational_PMS/PMDD_drugs
Class of receptors
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Gonadotropin_receptor
Chemical compound
but was subsequently discontinued. It seems to have been supplanted by relugolix (TAK-385), which is also under development by Takeda for the treatment
Sufugolix
Pharmaceutical drug
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Urofollitropin
Pharmaceutical drug
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Megestrol_acetate
Chemical compound
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Quadrosilan
Hormonal treatment for prostate cancer
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Androgen_deprivation_therapy
Chemical compound
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Ozarelix
Chemical compound
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Abarelix
Chemical compound
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Azagly-nafarelin
Teverelix (antarelix); Non-peptides: Elagolix Linzagolix Merigolix Opigolix Relugolix Sufugolix Gonadotropin LH/hCGTooltip Luteinizing hormone/choriogonadotropin
List of investigational sex-hormonal agents
List_of_investigational_sex-hormonal_agents
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
List_of_antiandrogens
Protein-coding gene in the species Homo sapiens
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Follicle-stimulating hormone receptor
Follicle-stimulating_hormone_receptor
Chemical compound
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Acyline
Pharmaceutical drug classification
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
ATC_code_G03
Chemical compound
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Fertirelin
Chemical compound
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Paroxypropione
Chemical compound
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Lecirelin
Chemical compound
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Metallibure
Chemical compound
Teverelix (antarelix); Non-peptides: Elagolix Linzagolix Merigolix Opigolix Relugolix Sufugolix Gonadotropin LH/hCGTooltip Luteinizing hormone/choriogonadotropin
Zoptarelin_doxorubicin
Chemical compound
Abarelix Cetrorelix Degarelix Ganirelix Non-peptide: Elagolix Linzagolix† Relugolix (+estradiol/norethisterone acetate) Gonadotropins Preparations Follicle-stimulating
Peforelin
RELUGOLIX
RELUGOLIX
RELUGOLIX
RELUGOLIX
Male
Hebrew
Variant spelling of Hebrew Yowshaphat, YOSHAFAT means "God has judged" or "whom God judges."Â
Boy/Male
Muslim
Poet, Knowledgeable
Boy/Male
Hindu
Love, Affection
Girl/Female
Latin
Honor.
Girl/Female
Hindu, Indian, Newdelhi, Tamil, Telugu
Silence; God
Boy/Male
Indian, Modern, Punjabi, Sikh
Embodiment of Beauty
Boy/Male
Celtic, Danish, French, German, Irish, Latin
Small and Mighty; To Rise Again; Small but Strong
Surname or Lastname
English
English : unexplained. Probably a habitational name from a lost or unidentified place.
Girl/Female
American, Christian, French, Indian
Dear or Beloved
Boy/Male
Bengali, Hindu, Indian, Punjabi, Sikh
The Lord Sun
RELUGOLIX
RELUGOLIX
RELUGOLIX
RELUGOLIX
RELUGOLIX