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BEDAQUILINE

  • Bedaquiline
  • Medication used to treat tuberculosis

    Bedaquiline, sometimes abbreviated as BDQ and sold under the brand name Sirturo, is a medication used for the treatment of active tuberculosis. Specifically

    Bedaquiline

    Bedaquiline

    Bedaquiline

  • Sorfequiline
  • Investigational drug

    generation diarylquinoline mycobacterial ATP synthase inhibitor. Compared to bedaquiline, it is claimed to have greater potency and reduced cardiac QT prolongation

    Sorfequiline

    Sorfequiline

    Sorfequiline

  • Pretomanid
  • Chemical compound

    tuberculosis affecting the lungs. It is generally used together with bedaquiline and linezolid. It is taken by mouth. The most common side effects include

    Pretomanid

    Pretomanid

    Pretomanid

  • Anil Koul
  • Indian scientist (born 1972)

    key role in the discovery and development of a new tuberculosis drug, bedaquiline, the first drug approved in 45 years for treatment of drug-resistant

    Anil Koul

    Anil Koul

    Anil_Koul

  • Diarylquinoline
  • Class of bacteria

    bacterial ATP synthase inhibition is an attractive therapeutic target. Bedaquiline (previously TMC207) is a 1,4-diaryl quinoline (phenyl and naphthyl).

    Diarylquinoline

    Diarylquinoline

    Diarylquinoline

  • Shreya Tripathi
  • Indian health activist (died 2018)

    to a respiratory disease center in New Delhi in the hopes of getting bedaquiline, a newly developed medication for XDR-TB. She was refused because she

    Shreya Tripathi

    Shreya_Tripathi

  • Tuberculosis
  • Infectious disease

    the acronyms BPaLM and BDLLfx: BPaLM (bedaquiline, pretomanid, linezolid, moxifloxacin). BDLLfxC (bedaquiline, delamanid, and linezolid in combination

    Tuberculosis

    Tuberculosis

    Tuberculosis

  • Everything Is Tuberculosis
  • 2025 nonfiction book by John Green

    Johnson & Johnson and Cepheid to ease access to the tuberculosis treatment bedaquiline and rapid diagnostic testing for multidrug-resistant tuberculosis, respectively

    Everything Is Tuberculosis

    Everything_Is_Tuberculosis

  • Timeline of antibiotics
  • first lipoglycopeptide 2010 – ceftaroline 2011 – fidaxomicin 2012 – bedaquiline 2013 – telavancin 2014 – tedizolid 2014 – dalbavancin 2014 – ceftolozane/tazobactam

    Timeline of antibiotics

    Timeline_of_antibiotics

  • Extensively drug-resistant tuberculosis
  • Tuberculosis that is resistant to the most effective drugs

    Administration (FDA) approved the use of pretomanid in combination with bedaquiline and linezolid for treating a limited and specific population of adult

    Extensively drug-resistant tuberculosis

    Extensively drug-resistant tuberculosis

    Extensively_drug-resistant_tuberculosis

  • Multidrug-resistant tuberculosis
  • Medical condition

    second-line TB drug groups: fluoroquinolones (moxifloxacin, ofloxacin), bedaquiline, linezolid, and injectable aminoglycosides (amikacin, streptomycin).

    Multidrug-resistant tuberculosis

    Multidrug-resistant tuberculosis

    Multidrug-resistant_tuberculosis

  • John Green
  • American author and YouTuber (born 1977)

    Johnson & Johnson (J&J) to allow generic versions of the tuberculosis drug bedaquiline to be produced, allowing increased global access to the drug. In May

    John Green

    John Green

    John_Green

  • Johnson & Johnson
  • American multinational pharmaceutical and medical device company

    Anti-Tuberculosis Drug Bedaquiline Rejected". The Wire. March 23, 2023. "Global Drug Facility Update on Access to Bedaquiline". Stop TB Partnership. July

    Johnson & Johnson

    Johnson & Johnson

    Johnson_&_Johnson

  • Propranolol
  • Beta blocker drug

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Propranolol

    Propranolol

    Propranolol

  • Gabapentin
  • Gamma-aminobutyric acid analog

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Gabapentin

    Gabapentin

    Gabapentin

  • Etripamil
  • Medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Etripamil

    Etripamil

  • Barbiturate
  • Class of depressant drugs derived from barbituric acid

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Barbiturate

    Barbiturate

    Barbiturate

  • Mycobacterium smegmatis
  • Species of bacterium

    second-line antitubercular drugs—including isoniazid, rifampicin, and bedaquiline—does not significantly increase the mutation rate. Instead, mycobacteria

    Mycobacterium smegmatis

    Mycobacterium smegmatis

    Mycobacterium_smegmatis

  • Biological half-life
  • Time taken for a drug to halve its concentration in blood plasma

    Österreichischer Apothekerverlag. Avodart 0,5 mg Weichkapseln. "Sirturo (bedaquiline) Tablets. Full Prescribing Information" (PDF). Janssen Products, Dec

    Biological half-life

    Biological half-life

    Biological_half-life

  • Calcium channel blocker
  • Drugs that disrupt movement of calcium across calcium channels

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Calcium channel blocker

    Calcium_channel_blocker

  • Ranolazine
  • Drug used to treat angina

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Ranolazine

    Ranolazine

    Ranolazine

  • Mycobacterium tuberculosis
  • Bacterium that causes tuberculosis

    Galik N, Toth J, Hirmondo R (15 November 2024). "Assessing the Impact of Bedaquiline, Clofazimine, and Linezolid on Mycobacterial Genome Integrity". Biomolecules

    Mycobacterium tuberculosis

    Mycobacterium tuberculosis

    Mycobacterium_tuberculosis

  • Lidocaine
  • Local anesthetic

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Lidocaine

    Lidocaine

    Lidocaine

  • Koen Andries
  • Belgian scientist

    discovery about a new di-Aryl-Quinoline-based drug (R207910), now called bedaquiline, which promises a shorter and simpler treatment for drug resistant Tuberculosis

    Koen Andries

    Koen_Andries

  • Antimicrobial resistance
  • Resistance of microbes to drugs directed against them

    Galik N, Toth J, Hirmondo R (15 November 2024). "Assessing the Impact of Bedaquiline, Clofazimine, and Linezolid on Mycobacterial Genome Integrity". Biomolecules

    Antimicrobial resistance

    Antimicrobial resistance

    Antimicrobial_resistance

  • Cocaine
  • Tropane alkaloid and stimulant drug

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Cocaine

    Cocaine

    Cocaine

  • Erythromycin
  • Antibiotic medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Erythromycin

    Erythromycin

    Erythromycin

  • Phenytoin
  • Anti-seizure medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Phenytoin

    Phenytoin

    Phenytoin

  • Amlodipine
  • Medication against high blood pressure

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Amlodipine

    Amlodipine

    Amlodipine

  • Rhynchophylline
  • Chemical compound

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Rhynchophylline

    Rhynchophylline

    Rhynchophylline

  • CB03-154
  • Pharmaceutical compound

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    CB03-154

    CB03-154

    CB03-154

  • Amitriptyline
  • Tricyclic antidepressant

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Amitriptyline

    Amitriptyline

    Amitriptyline

  • Doxepin
  • Sedating antidepressant

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Doxepin

    Doxepin

    Doxepin

  • Chlorpromazine
  • Typical antipsychotic medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Chlorpromazine

    Chlorpromazine

    Chlorpromazine

  • Lorazepam
  • Benzodiazepine medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Lorazepam

    Lorazepam

    Lorazepam

  • Ketamine
  • Dissociative anesthetic and anti-depressant

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Ketamine

    Ketamine

    Ketamine

  • Sotalol
  • Medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Sotalol

    Sotalol

    Sotalol

  • Michael Niederweis
  • Professor of Microbiology

    "Molecular structure determined for efflux pumps that confer tuberculosis bedaquiline resistance". www.uab.edu. Retrieved 2025-10-20. Jackson, Mary; Stevens

    Michael Niederweis

    Michael Niederweis

    Michael_Niederweis

  • WHO Model List of Essential Medicines
  • Formulary by the World Health Organization

    Amikacin Amoxicillin/clavulanic acid (amoxicillin + clavulanic acid) Bedaquiline Clofazimine Cycloserine Delamanid Ethambutol Ethambutol/isoniazid/py

    WHO Model List of Essential Medicines

    WHO_Model_List_of_Essential_Medicines

  • Kava
  • Species of plant

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Kava

    Kava

    Kava

  • Mirogabalin
  • Chemical compound

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Mirogabalin

    Mirogabalin

    Mirogabalin

  • Lamotrigine
  • Anticonvulsant medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Lamotrigine

    Lamotrigine

    Lamotrigine

  • Meclizine
  • Chemical compound

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Meclizine

    Meclizine

    Meclizine

  • Nifedipine
  • Calcium channel blocker medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Nifedipine

    Nifedipine

    Nifedipine

  • Diltiazem
  • Calcium channel blocker medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Diltiazem

    Diltiazem

    Diltiazem

  • Nicorandil
  • Chemical compound

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Nicorandil

    Nicorandil

    Nicorandil

  • Suzetrigine
  • Non-opioid analgesic drug

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Suzetrigine

    Suzetrigine

    Suzetrigine

  • Baclofen
  • Muscle relaxant medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Baclofen

    Baclofen

    Baclofen

  • Janssen Pharmaceuticals
  • Belgian pharmaceutical company

    Nizoral (ketoconazole) (Removed in 2005) Risperdal (risperidone) Sirturo (bedaquiline) – an diarylquinoline anti-tuberculosis drug, discovered by Koen Andries

    Janssen Pharmaceuticals

    Janssen_Pharmaceuticals

  • G protein-coupled inwardly rectifying potassium channel
  • Family of ion channels

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    G protein-coupled inwardly rectifying potassium channel

    G_protein-coupled_inwardly_rectifying_potassium_channel

  • Nicardipine
  • Antihypertensive drug of the calcium channel blocker class

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Nicardipine

    Nicardipine

    Nicardipine

  • Astemizole
  • Antihistamine drug

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Astemizole

    Astemizole

    Astemizole

  • Phenibut
  • CNS depressant medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Phenibut

    Phenibut

    Phenibut

  • Ketoconazole
  • Antifungal chemical compound

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Ketoconazole

    Ketoconazole

    Ketoconazole

  • ATC code J04
  • Pharmaceutical drug classification

    Pyrazinamide J04AK02 Ethambutol J04AK03 Terizidone J04AK04 Morinamide J04AK05 Bedaquiline J04AK06 Delamanid J04AK07 Amithiozone J04AK08 Pretomanid J04AM01 Streptomycin

    ATC code J04

    ATC_code_J04

  • Safinamide
  • Reversible monoamine oxidase B inhibitor

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Safinamide

    Safinamide

    Safinamide

  • Pynegabine
  • Pharmaceutical compound

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Pynegabine

    Pynegabine

    Pynegabine

  • Procaine
  • Local anesthetic drug

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Procaine

    Procaine

    Procaine

  • Carbamazepine
  • Anticonvulsant medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Carbamazepine

    Carbamazepine

    Carbamazepine

  • Benzocaine
  • Local anaesthetic drug

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Benzocaine

    Benzocaine

    Benzocaine

  • Sodium channel
  • Transmembrane protein allowing sodium ions in and out

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Sodium channel

    Sodium channel

    Sodium_channel

  • Pethidine
  • Opioid analgesic

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Pethidine

    Pethidine

    Pethidine

  • Mefenamic acid
  • Chemical compound

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Mefenamic acid

    Mefenamic acid

    Mefenamic_acid

  • Quabodepistat
  • Pharmaceutical compound

    et al. (January 2024). "Quabodepistat in combination with delamanid and bedaquiline in participants with drug-susceptible pulmonary tuberculosis: protocol

    Quabodepistat

    Quabodepistat

    Quabodepistat

  • Vanoxerine
  • Chemical compound

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Vanoxerine

    Vanoxerine

    Vanoxerine

  • Phumeza Tisile
  • South African tuberculosis activist

    advocated for patient access to XDR-TB drugs including linezolid and bedaquiline. Tisile's successful treatment relied on linezolid, which was expensive

    Phumeza Tisile

    Phumeza_Tisile

  • Ion channel
  • Pore-forming membrane protein

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Ion channel

    Ion channel

    Ion_channel

  • Anand Grover
  • Indian lawyer

    Grover represented Shreya Tripathi in her successful efforts to obtain bedaquiline for the treatment of her extensively drug-resistant tuberculosis. Grover

    Anand Grover

    Anand_Grover

  • Diphenhydramine
  • Antihistamine medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Diphenhydramine

    Diphenhydramine

    Diphenhydramine

  • Leconotide
  • Conotoxin peptide under investigation as an analgesic drug

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Leconotide

    Leconotide

  • Neglected tropical diseases
  • Diverse group of tropical infectious diseases which are common in developing countries

    NTD PRVs to date (December 2014): Coartem (by Novartis, for malaria); bedaquiline (by Janssen, for TB); and miltefosine (by Knight, for leishmaniasis)

    Neglected tropical diseases

    Neglected tropical diseases

    Neglected_tropical_diseases

  • Topiramate
  • Medication used to treat epilepsy and migraine

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Topiramate

    Topiramate

    Topiramate

  • Haloperidol
  • Typical antipsychotic medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Haloperidol

    Haloperidol

    Haloperidol

  • Benzonatate
  • Oral cough medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Benzonatate

    Benzonatate

  • Nortriptyline
  • Antidepressant medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Nortriptyline

    Nortriptyline

    Nortriptyline

  • Atomoxetine
  • Medication used to treat ADHD

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Atomoxetine

    Atomoxetine

    Atomoxetine

  • Cyproheptadine
  • Antihistamine medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Cyproheptadine

    Cyproheptadine

    Cyproheptadine

  • XOB
  • Pharmaceutical compound

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    XOB

    XOB

  • Dextropropoxyphene
  • Withdrawn opioid medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Dextropropoxyphene

    Dextropropoxyphene

    Dextropropoxyphene

  • Ajmaline
  • Chemical compound

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Ajmaline

    Ajmaline

    Ajmaline

  • Bretylium
  • Chemical compound

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Bretylium

    Bretylium

    Bretylium

  • Fostedil
  • Chemical compound

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Fostedil

    Fostedil

    Fostedil

  • Crisugabalin
  • Drug for chronic pain

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Crisugabalin

    Crisugabalin

    Crisugabalin

  • Chlorphenamine
  • Antihistamine used to treat allergies

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Chlorphenamine

    Chlorphenamine

    Chlorphenamine

  • Sodium channel blocker
  • Several medications which disrupt the movement of Na+ ions

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Sodium channel blocker

    Sodium_channel_blocker

  • Tetrodotoxin
  • Neurotoxin

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Tetrodotoxin

    Tetrodotoxin

    Tetrodotoxin

  • Buprenorphine
  • Opioid used to treat pain and opioid use disorder

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Buprenorphine

    Buprenorphine

    Buprenorphine

  • Terfenadine
  • Chemical compound

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Terfenadine

    Terfenadine

    Terfenadine

  • Tetrandrine
  • Chemical compound

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Tetrandrine

    Tetrandrine

    Tetrandrine

  • Delamanid
  • Chemical compound

    globally as of 2015. It was believed that pricing will be similar to bedaquiline, which for six months is approximately US$900 in low income countries

    Delamanid

    Delamanid

  • Promethazine
  • Sedating antihistamine

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Promethazine

    Promethazine

    Promethazine

  • Valproate
  • Medication used for epilepsy, bipolar disorder and migraine

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Valproate

    Valproate

    Valproate

  • Clofazimine
  • Medication

    resistant tuberculosis in combination with other second-line agents such as bedaquiline. Other uses have not been proven to be safe or effective. It has been

    Clofazimine

    Clofazimine

    Clofazimine

  • Aliskiren/amlodipine/hydrochlorothiazide
  • Pharmaceutical drug

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Aliskiren/amlodipine/hydrochlorothiazide

    Aliskiren/amlodipine/hydrochlorothiazide

  • Alcohol (drug)
  • Active ingredient in fermented drinks

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Alcohol (drug)

    Alcohol (drug)

    Alcohol_(drug)

  • VSN16R
  • Pharmaceutical compound

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    VSN16R

    VSN16R

    VSN16R

  • Azetukalner
  • Experimental anticonvulsant

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Azetukalner

    Azetukalner

    Azetukalner

  • Solifenacin
  • Chemical compound

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Solifenacin

    Solifenacin

    Solifenacin

  • Pregabalin
  • Anticonvulsant medication

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Pregabalin

    Pregabalin

    Pregabalin

  • Funapide
  • Analgesic drug under development

    Ajmaline Amiodarone AmmTX3 Astemizole Azaspiracid AZD1305 Azimilide Bedaquiline BeKm-1 BmTx3 BRL-32872 Chlorpromazine Cisapride Clarithromycin Darifenacin

    Funapide

    Funapide

    Funapide

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