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Chemical compound
Carbidopa, sold under the brand name Lodosyn, is a medication used primarily in the treatment of Parkinson's disease. A DOPA decarboxylase inhibitor,
Carbidopa
Parkinson's disease medication
Carbidopa/levodopa, sold under the brand name Sinemet among others, is a fixed-dose combination used for the treatment of Parkinson's disease. It contains
Carbidopa/levodopa
Parkinson's disease medication
Carbidopa/levodopa/entacapone, sold under the brand name Stalevo among others, is a dopaminergic fixed-dose combination medication that contains carbidopa
Carbidopa/levodopa/entacapone
Chemical compound
treatment of Parkinson's disease. Entacapone together with levodopa and carbidopa allows levodopa to have a longer effect in the brain and reduces Parkinson's
Entacapone
Dopaminergic medication
with carbidopa (as levodopa/carbidopa), with benserazide (as levodopa/benserazide), and with both carbidopa and entacapone (as levodopa/carbidopa/entacapone)
Levodopa
Combination dopaminergic medication
Melevodopa/carbidopa, sold under the brand name Sirio, is a combination of melevodopa, a prodrug of the dopamine precursor and hence non-selective dopamine
Melevodopa/carbidopa
Medication
Carbidopa/oxitriptan (developmental code name EVX-101), or carbidopa/5-hydroxytryptophan (carbidopa/5-HTP), is a combination of 5-hydroxytryptophan (5-HTP;
Carbidopa/oxitriptan
Combination medication
for carbidopa; and foslevodopa, an aromatic amino acid and prodrug for levodopa that was developed by AbbVie. Its structure is identical to carbidopa/levodopa
Foscarbidopa/foslevodopa
Chemical compound
such as carbidopa or benserazide. These agents increase the strength and duration of levodopa. Combination formulations include levodopa/carbidopa and levodopa/benserazide
L-DOPA
OTC medication for depression
between the seven studies examined. At high doses, or in combination with carbidopa, 5-HTP has been used to treat obesity (by promoting weight loss). MDMA
Oxitriptan
Chemical compound
Foscarbidopa is a medication which acts as a prodrug for carbidopa. It is used in a subcutaneous infusion as a fixed-dose combination with foslevodopa
Foscarbidopa
Chemical compound
water solubility of tablet levodopa. In combination with carbidopa, as melevodopa/carbidopa (brand name Sirio), it is approved for use in the treatment
Melevodopa
Investigational Parkinson's disease drugs
diagnosis [1] Levodopa/carbidopa subcutaneous (ND-0612; ND-0680) – combination of levodopa (dopamine precursor) and carbidopa (aromatic L-amino acid decarboxylase
List of investigational Parkinson's disease drugs
List_of_investigational_Parkinson's_disease_drugs
Syndrome characterized by tremor, slowed movements, rigidity, and imbalance
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Parkinsonism
Formulary by the World Health Organization
Cladribineα Glatiramer acetateα Rituximabα Biperiden Levodopa/carbidopa (levodopa + carbidopa) Baclofen Acetylsalicylic acid (aspirin) Ibuprofen Paracetamol
WHO Model List of Essential Medicines
WHO_Model_List_of_Essential_Medicines
Medication
with levodopa and an aromatic L-amino acid decarboxylase inhibitor (e.g. carbidopa or benserazide). The therapeutic benefit of using a COMT inhibitor is
Catechol-O-methyltransferase inhibitor
Catechol-O-methyltransferase_inhibitor
Canadian-American actor and activist (born 1961)
(PPMI). Fox manages the symptoms of his Parkinson's disease with the drug carbidopa/levodopa. He had a thalamotomy in 1998. In Lucky Man, Fox wrote that he
Michael_J._Fox
Progressive neurodegenerative disease
catechol-O-methyltransferase can cause nausea and vomiting; inhibitors such as carbidopa, entacapone, and benserazide are usually taken with levodopa to mitigate
Parkinson's_disease
Chemical compound
name Nourianz, is a medication used as an add-on treatment to levodopa/carbidopa in adults with Parkinson's disease (PD) experiencing "off" episodes. Istradefylline
Istradefylline
Compounds metabolized into monoamines
decarboxylase (DDC) inhibitors) such as carbidopa and benserazide to restrict metabolism and activation in the periphery. Carbidopa/levodopa and levodopa/benserazide
Monoamine_precursor
Chemical compound
In the US, opicapone is indicated as adjunctive treatment to levodopa/carbidopa in people with Parkinson's disease (PD) experiencing "off" episodes. The
Opicapone
Chemical compound
to levodopa/carbidopa or levodopa/benserazide medications. Levodopa is a prodrug for dopamine, which reduces Parkinson symptoms; carbidopa and benserazide
Tolcapone
Excess deposition of extracellular matrix in the cardiac muscle
5-HTP is also sold without carbidopa as a dietary supplement, and may have increased risks when taken by itself without carbidopa.[citation needed] Cardiac
Cardiac_fibrosis
Disorder of diminished motivation
as bromocriptine or amantadine. Other treatments include amantadine, carbidopa-levodopa, donepezil, memantine, and oral magnesium oxide. Fourteen-year-old
Akinetic_mutism
Medical condition
is currently being treated using a combination therapy of levodopa and carbidopa. These treatments are also used for individuals suffering from Parkinson's
Sepiapterin reductase deficiency
Sepiapterin_reductase_deficiency
Chemical compound often used as medication
Canada, both made by Roche. Benserazide is not approved for use in the US; carbidopa is used, instead, for the same purpose. These combinations are also used
Benserazide
Type of medication
blood–brain barrier. Examples of extracerebral decarboxylase inhibitors include carbidopa and benserazide. Peripherally selective DDCIs incapable of crossing the
Aromatic L-amino acid decarboxylase inhibitor
Aromatic_L-amino_acid_decarboxylase_inhibitor
Chemical compound
selective aromatic L-amino acid decarboxylase (AAAD) inhibitor such as carbidopa or benserazide. These agents increase the strength and duration of oxitriptan
5-Hydroxytryptophan
Parasympathetic nervous system inhibitors
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Anticholinergic
Slow mental activity
bradykinesia, could be treated using the combination of a L-DOPA and carbidopa regimen. This combination was believed to alter these effects of Parkinson's
Bradyphrenia
Synthetic amino acid/norepinephrine prodrug
decarboxylase inhibitor (AAADI) or DOPA decarboxylase inhibitor (DDC) such as carbidopa (Lodosyn) to increase central norepinephrine concentrations while minimizing
Droxidopa
Drug used to treat influenzavirus A infection
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Rimantadine
Involuntary movements of parts of the body
also a common presentation of dyskinesia as a side effect of levodopa-carbidopa in the treatment of Parkinson disease. The use of crack cocaine or amphetamines
Choreoathetosis
D1 receptor positive allosteric modulator under development for Parkinson's disease
D1 receptor, as well as approaches to sub-cutaneously deliver levodopa/carbidopa such as Abbvie's ABBV-951 and Neuroderm's ND0612. "Glovadalen". IUPHAR/BPS
Glovadalen
Biopharmaceutical company
of Parkinson's disease Vimpat (lacosamide), an anticonvulsant Atamet (carbidopa/levodopa) for Parkinson's disease Nayzilam (midazolam) for Seizure Clusters
UCB_(company)
Abandoned anticholinergic
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Benapryzine
Chemical compound
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Nitecapone
Medication
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Tavapadon
Chemical compound
4-dihydroxyphenylalanine (DFMD, DFM-DOPA) is a DOPA decarboxylase inhibitor. Carbidopa Methyldopa Zbinden G, Brändle E (February 1980). "Inhibition of 5-hydroxytryptophan
Α-Difluoromethyl-DOPA
Dopamine agonist medication
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Pramipexole
Abandoned antiparkinsonian agent
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Botiacrine
Medication
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Levodopa/benserazide
Psychological sensation
similar symptoms while taking a combination of 5-hydroxytryptophan and carbidopa. Déjà vu may happen if a person experienced the current sensory experience
Déjà_vu
Group of antidepressants
names indicate major drugs. Carbenzide Cimemoxin Domoxin Metfendrazine Carbidopa Centazolone López-Muñoz F, Alamo C (2009). "Monoaminergic neurotransmission:
Hydrazine_(antidepressant)
Investigational obsessive–compulsive disorder drugs
psychedelic hallucinogen [1] Carbidopa/oxytriptan (EVX-101; carbidopa/oxitriptan; carbidopa/5-HTP) – combination of carbidopa (aromatic L-amino-acid decarboxylase
List of investigational obsessive–compulsive disorder drugs
List_of_investigational_obsessive–compulsive_disorder_drugs
Antihistamine medication
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Diphenhydramine
Treatment of Parkinson's disease
portable pump Duodopa or Levodopa-carbidopa intestinal gel (LCIG), a methylcellulose-based suspension of levodopa and carbidopa delivered in a continuous way
Management of Parkinson's disease
Management_of_Parkinson's_disease
Group of stereoisomers
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Procyclidine
Medical condition from optic nerve damage
ischemia. Proposed treatments include hyperbaric oxygen, levodopa or carbidopa, aspirin, transvitreal optic neurotomy, bevacizumab and vitrectomy. The
Non-arteritic anterior ischemic optic neuropathy
Non-arteritic_anterior_ischemic_optic_neuropathy
Chemical compound
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Tigloidine
Class of prescription drugs in India
CALCIUM DOBESILATE 78. CANDESARTAN 79. CAPECITABINE 80. CAPTOPRIL 81. CARBIDOPA 82. CARBOCISTEINE 83. CARBOPLATIN 84. CARBOQUONE 85. CARISOPRODOL 86.
Schedule_H
Chemical compound
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Phenglutarimide
DMT-infused smoking blend
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
Changa_(drug)
Subtype of delusion
J-T Y.; Ziegler, D. (1976). "Psychiatric symptoms with initiation of carbidopa-levodopa treatment". Neurology. 26 (7): 679–700. doi:10.1212/wnl.26.7
Delusions_of_grandeur
Chemical compound
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
3-Hydroxymorphinan
Organic chemical that functions both as a hormone and a neurotransmitter
co-administered with an enzyme inhibitor of peripheral decarboxylation such as carbidopa or benserazide, to reduce the amount converted to dopamine in the periphery
Dopamine
Skeletal muscle relaxant
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Orphenadrine
Experimental enzyme inhibitor
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
Vafidemstat
Dopamine agonist medication
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Piribedil
Pharmaceutical compound
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
Sembragiline
Pharmaceutical drug classification
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
ATC_code_N04
Medication for movement disorders
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Benzatropine
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
LBT-3627
Medication
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Rasagiline
Chemical compound
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Lazabemide
Class of enzymes
mild depression or dysthymia).[citation needed] AADC is inhibited by carbidopa outside of the blood brain barrier to inhibit the premature conversion
Aromatic L-amino acid decarboxylase
Aromatic_L-amino_acid_decarboxylase
Chemical compound
therapy, together with levodopa and a decarboxylase inhibitor such as carbidopa, in progressive-phase Parkinson's disease; In some countries also: ablactation
Cabergoline
Experimental antiparkinsonian agent and adamantane derivative
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
Hemantane
Pharmaceutical compound
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
Tisolagiline
3-Iodotyrosine • Aquayamycin • Bulbocapnine • Metirosine • Oudenone Benserazide • Carbidopa • Genistein • Methyldopa Nonselective: Benmoxin • Caroxazone • Echinopsidine •
List_of_dopaminergic_drugs
Antispasmodic drug
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Trihexyphenidyl
Anti-hypertension medication
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
Hydralazine
Chemical compound
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
Carnegine
Drug that binds to but does not activate muscarinic cholinergic receptors
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Muscarinic_antagonist
COMT inhibitor
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
Neluxicapone
Chemical compound
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Apomorphine
Dopamine agonist medication
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Ropinirole
Class of enzymes
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
Phenylethanolamine N-methyltransferase
Phenylethanolamine_N-methyltransferase
Pharmaceutical compound
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
Tryptoline
Chemical compound
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
Disulfiram
Chemical compound
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
Furazolidone
Chemical compound
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Bornaprine
Blue dye also used as a medication
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
Methylene_blue
Medication used to treat high blood pressure
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Methyldopa
3-Iodotyrosine Aquayamycin Bulbocapnine Metirosine Oudenone Benserazide Carbidopa Genistein Methyldopa Bupicomide Disulfiram Dopastin Fusaric acid Nepicastat
List_of_adrenergic_drugs
South American psychoactive decoction
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
Ayahuasca
MAOI antidepressant
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
Encyprate
Medication used to treat Alzheimer's disease
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Memantine
Pharmaceutical compound
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
6-Methoxyharmalan
Human development following adolescence
Suneel (April 2013). "Extended-release carbidopa-levodopa (IPX066) compared with immediate-release carbidopa-levodopa in patients with Parkinson's disease
Adult_development
Chemical compound
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Piroheptine
Chemical compound
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Aplindore
American biotechnology company
of off episodes in patients with Parkinson's disease currently taking carbidopa/levodopa. Inbrija is approved by the FDA and the EU. BTT1023 (timolumab)
Acorda_Therapeutics
Chemical compound
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
5-MAPBT
Pharmaceutical compound
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
3,4-Dimethoxyamphetamine
Chemical compound
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
Α-Methyl-p-tyrosine
Group of stereoisomers
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Biperiden
Chemical compound
precursors Levodopa# (+benserazide, +carbidopa, +carbidopa/entacapone) Foslevodopa (+foscarbodipa) Melevodopa (+carbidopa) DA receptor agonists Ergoline: Bromocriptine
Foslevodopa
American publicly traded generics and specialty pharmaceutical company
Amneal filed for FDA approval of a new specialty drug labeled IPX-203, (carbidopa-levodopa) which is designed to help control symptoms in Parkinson's disease
Amneal_Pharmaceuticals
Agricultural product processed from the leaves of plants in the genus Nicotiana
L-Tyrosine→Tyramine Tryptophan→Tryptamine Inhibitors: Benserazide Carbidopa DFMD Genistein Methyldopa MAOTooltip Monoamine oxidase Substrates→Products
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