Search references for ALLOSTERIC SEROTONIN-REUPTAKE-INHIBITOR. Phrases containing ALLOSTERIC SEROTONIN-REUPTAKE-INHIBITOR
See searches and references containing ALLOSTERIC SEROTONIN-REUPTAKE-INHIBITOR!ALLOSTERIC SEROTONIN-REUPTAKE-INHIBITOR
Class of drug
A serotonin reuptake inhibitor (SRI) is a type of drug which acts as a reuptake inhibitor of the neurotransmitter serotonin (5-hydroxytryptamine, or 5-HT)
Serotonin_reuptake_inhibitor
Allosteric serotonin reuptake inhibitor is a type of selective serotonin reuptake inhibitor (SSRI). Evidence of the allosteric action of escitalopram on
Allosteric serotonin reuptake inhibitor
Allosteric_serotonin_reuptake_inhibitor
Class of drug
Serotonin antagonist and reuptake inhibitors (SARIs) are a class of drugs used mainly as antidepressants, but also as anxiolytics and hypnotics. They act
Serotonin antagonist and reuptake inhibitor
Serotonin_antagonist_and_reuptake_inhibitor
Class of antidepressant medication
Serotonin–norepinephrine reuptake inhibitors (SNRIs) are a class of antidepressant medications used to treat major depressive disorder (MDD), anxiety disorders
Serotonin–norepinephrine reuptake inhibitor
Serotonin–norepinephrine_reuptake_inhibitor
Class of drugs
A serotonin–norepinephrine–dopamine reuptake inhibitor (SNDRI), also known as a triple reuptake inhibitor (TRI or TUI), is a type of drug that acts as
Serotonin–norepinephrine–dopamine reuptake inhibitor
Serotonin–norepinephrine–dopamine_reuptake_inhibitor
Medications that increase norepinephrine
A norepinephrine reuptake inhibitor (NRI), also known as a noradrenaline reuptake inhibitor or adrenergic reuptake inhibitor, is a type of drug that acts
Norepinephrine reuptake inhibitor
Norepinephrine_reuptake_inhibitor
Class of antidepressant medication
serotonin neurotransmitter system. To be precise, SMSs simultaneously modulate one or more serotonin receptors and inhibit the reuptake of serotonin.
Serotonin modulator and stimulator
Serotonin_modulator_and_stimulator
Class of antidepressant medication
Selective serotonin reuptake inhibitors (SSRIs) are a class of drugs that are typically used as antidepressants in the treatment of major depressive disorder
Selective serotonin reuptake inhibitor
Selective_serotonin_reuptake_inhibitor
Drug that inhibits the reuptake of norepinephrine and dopamine
A norepinephrine–dopamine reuptake inhibitor (NDRI) is a type of drug that inhibits the reuptake of the monoamine neurotransmitters norepinephrine and
Norepinephrine–dopamine reuptake inhibitor
Norepinephrine–dopamine_reuptake_inhibitor
SSRI antidepressant
among others, is an antidepressant medication of the selective serotonin reuptake inhibitor (SSRI) class used for the treatment of major depressive disorder
Fluoxetine
SSRI antidepressant
among others, is an antidepressant medication of the selective serotonin reuptake inhibitor (SSRI) class. It is mainly used to treat major depressive disorder
Escitalopram
SSRI antidepressant
among others, is an antidepressant medication of the selective serotonin reuptake inhibitor (SSRI) class used to treat major depressive disorder, generalized
Sertraline
Type of drug
reuptake inhibitor Monoamine reuptake inhibitor Dopamine reuptake inhibitor Norepinephrine reuptake inhibitor Serotonin reuptake inhibitor Serotonin-norepinephrine
Reuptake_inhibitor
Mammalian protein found in humans
of serotonin to transporters (serotonin reuptake inhibitors, or SRIs) are used to treat mental disorders. The selective serotonin reuptake inhibitor (SSRI)
Serotonin_transporter
Type of medication
treatments, including selective serotonin reuptake inhibitors (SSRIs), serotonin–norepinephrine reuptake inhibitors (SNRIs), mirtazapine, bupropion,
Monoamine_oxidase_inhibitor
Medication mainly used for depression and smoking cessation
the cases of "incomplete response" to the first-line selective serotonin reuptake inhibitor (SSRI) antidepressant. Bupropion has several features that distinguish
Bupropion
Serotonin modulator antidepressant
class of serotonin modulators and stimulators, which also includes vilazodone. More specifically, vortioxetine is a serotonin reuptake inhibitor, agonist
Vortioxetine
Class of drug
A dopamine reuptake inhibitor (DRI) is a class of drug which acts as a reuptake inhibitor of the monoamine neurotransmitter dopamine by blocking the action
Dopamine_reuptake_inhibitor
Drug class
An adenosine reuptake inhibitor (AdoRI) is a type of drug which acts as a reuptake inhibitor for the purine nucleoside and neurotransmitter adenosine
Adenosine_reuptake_inhibitor
SNRI antidepressant
among others, is an antidepressant medication of the serotonin–norepinephrine reuptake inhibitor (SNRI) class. It is used to treat major depressive disorder
Venlafaxine
Antidepressant medication
a strong norepinephrine reuptake inhibitor and a moderate serotonin reuptake inhibitor. Additionally, nortriptyline inhibits the activity of histamine
Nortriptyline
SSRI antidepressant
name Luvox among others, is an antidepressant of the selective serotonin reuptake inhibitor (SSRI) class. It is primarily used to treat major depressive
Fluvoxamine
Antiretroviral medication
dual GABAA receptor positive allosteric modulator and orthosteric site antagonist, as a serotonin–dopamine reuptake inhibitor (SDRI), as a vesicular monoamine
Efavirenz
Antidepressant
relatively selective norepinephrine reuptake inhibitor, though it does also have other activities such as weak serotonin reuptake inhibitory, α1-blocking, antihistamine
Desipramine
SSRI antidepressant
among others, is an antidepressant medication of the selective serotonin reuptake inhibitor (SSRI) class used to treat major depressive disorder, obsessive–compulsive
Paroxetine
Tricyclic antidepressant medication
a norepinephrine reuptake inhibitor but a stronger serotonin reuptake inhibitor and helps to balance amoxapine's ratio of serotonin to norepinephrine
Amoxapine
SSRI antidepressant
name Celexa among others, is an antidepressant of the selective serotonin reuptake inhibitor (SSRI) class. It is used to treat major depressive disorder,
Citalopram
Antidepressant medication
Mirtazapine in combination with a selective serotonin reuptake inhibitor, serotonin–norepinephrine reuptake inhibitor, or tricyclic antidepressant as an augmentation
Mirtazapine
Chemical compound
inhibitor of monoamine oxidase A (RIMA), but it also inhibits the reuptake of serotonin. THH contributes to B. caapi's psychoactivity as a serotonin reuptake
Tetrahydroharmine
Antidepressant medication
recommended. It is in the serotonin modulator class of medications and is believed to work both as a selective serotonin reuptake inhibitor (SSRI) and activator
Vilazodone
Class of compounds
relative to the selective serotonin reuptake inhibitors (SSRIs). A closely related type of drug is a serotonin reuptake inhibitor (SRI), for instance fluoxetine
Serotonin_releasing_agent
Tricyclic antidepressant
As with other antidepressants (notably including selective serotonin reuptake inhibitors), it may paradoxically increase the risk of suicide in those
Clomipramine
Synthetic opioid pain medication
Tramal among others, is an opioid pain medication and a serotonin–norepinephrine reuptake inhibitor (SNRI) used to treat moderate to severe pain. When taken
Tramadol
Group of chemical compounds
including DNA mutagenic effects, imidazoline receptor interactions, serotonin reuptake inhibition, monoamine oxidase inhibition, cytochrome P450 enzyme inhibition
Β-Carboline
(Viibryd) – serotonin 5-HT1A receptor partial agonist and serotonin reuptake inhibitor SNTX-2643 (SENS-01) – atypical serotonin reuptake inhibitor (SRI) (kanna-derived)
List of investigational social anxiety disorder drugs
List_of_investigational_social_anxiety_disorder_drugs
Antidepressant medication
and insomnia. It is a phenylpiperazine compound of the serotonin antagonist and reuptake inhibitor (SARI) class. The medication is taken orally. Common
Trazodone
Sedating antidepressant
as an inhibitor of serotonin and norepinephrine reuptake than (E)-doxepin. The selectivity of doxepin for inhibition of norepinephrine reuptake over that
Doxepin
Drug that makes neurotransmitter transporters more active
was once claimed to be a (selective) serotonin reuptake enhancer (SRE or SSRE), but the role of serotonin reuptake in its mechanism is doubtful. Tianeptine
Reuptake_enhancer
Medication used to treat ADHD
sold under the brand name Strattera, is a selective norepinephrine reuptake inhibitor (SNRI) medication used to treat attention deficit hyperactivity disorder
Atomoxetine
Antidepressant
effects on: Serotonin: very strong reuptake inhibition. Imipramine is a tertiary TCA, and is a potent inhibitor of serotonin reuptake, and to a greater
Imipramine
Class of medications used to alleviate anxiety
The first serotonin norepinephrine reuptake inhibitor (SNRI), venlafaxine (Effexor), entered the market in 1993. SNRIs can target serotonin and norepinephrine
Anxiolytic
Muscle relaxant medication
is unclear. In any case, it is known to inhibit serotonin and norepinephrine reuptake and to block serotonin, adrenergic, histamine, and muscarinic acetylcholine
Cyclobenzaprine
Investigational PTSD drugs
Serestill) – selective serotonin reuptake inhibitor (SSRI) [64] [65] Sertraline (Lustral, Zoloft) – selective serotonin reuptake inhibitor (SSRI) [66] Antipsychotics
List of investigational post-traumatic stress disorder drugs
List_of_investigational_post-traumatic_stress_disorder_drugs
Investigational generalized anxiety disorder drugs
Ruoxinlin) – serotonin–norepinephrine–dopamine reuptake inhibitor (SNDRI) [4] Vilazodone (EMD-68843; SB-659746A; Viibryd) – serotonin reuptake inhibitor (SRI)
List of investigational generalized anxiety disorder drugs
List_of_investigational_generalized_anxiety_disorder_drugs
Active metabolite of paracetamol
same way that common selective serotonin reuptake inhibitor (SSRI) antidepressants prevent the reuptake of serotonin. Earlier work on the mechanism of
AM404
Pharmaceutical compound
DMHT is a potent serotonin reuptake inhibitor (SRI), with an affinity (IC50Tooltip half-maximal inhibitory concentration) for the serotonin transporter (SERT)
Dimethylhomotryptamine
SNRI medication
sold under the brand name Savella among others, is a serotonin–norepinephrine reuptake inhibitor (SNRI) used in the clinical treatment of fibromyalgia
Milnacipran
Chemical compound
antagonist and also a triple reuptake inhibitor which inhibits reuptake of all three monoamine neurotransmitters serotonin, dopamine and noradrenaline
3-Methyl-PCPy
Withdrawn atypical antidepressant drug
preferentially as a relatively weak dopamine reuptake inhibitor, but also as an even weaker serotonin reuptake inhibitor (IC50 = 1,500 nM) and as a weak antagonist
Medifoxamine
Monoamine neurotransmitter
antidepressants, including selective serotonin reuptake inhibitors (SSRIs) and serotonin–norepinephrine reuptake inhibitors (SNRIs), which block reabsorption
Serotonin
Trevilor) Serotonin–dopamine reuptake inhibitors include: None currently marketed Medifoxamine (Clédial, Gerdaxy) Serotonin–norepinephrine–dopamine reuptake inhibitors
List_of_antidepressants
Antidepressant
therapeutic advantages over other TCAs. It acts as a serotonin–norepinephrine reuptake inhibitor (SNRI) and also has other activities including antihistamine
Dosulepin
Cough suppressant and dissociative drug
mechanisms of action, including actions as a nonselective serotonin–norepinephrine reuptake inhibitor and a sigma-1 receptor agonist. Dextromethorphan and
Dextromethorphan
Pharmaceutical compound
known as N-desalkylquetiapine, is a 5-HT2B serotonin receptor modulator, and norepinephrine reuptake inhibitor. It is the principal metabolite of quetiapine
Norquetiapine
Appetite suppressant
suppressants, mazindol is thought to act as a reuptake inhibitor of norepinephrine, dopamine, and serotonin. In addition to its other actions, mazindol
Mazindol
Pharmaceutical compound
not of the serotonin 5-HT1A receptor. It is also a serotonin–norepinephrine–dopamine reuptake inhibitor (SNDRI). The chemical synthesis of PALT has been
Propylallyltryptamine
Substituted cathinone stimulant drug
transporter) and 383 nM (serotonin transporter). The methylenedioxy ring-substitution provides a higher potency at inhibiting serotonin reuptake than its analogue
N-Ethylpentylone
Chemical compound
nefazodone, and may contribute significantly to its effects. Serotonin antagonist and reuptake inhibitor Golden RN, Dawkins K, Nicholas L (2017). "Trazodone and
Hydroxynefazodone
Subtype of serotonin receptor
selective serotonin reuptake inhibitors (SSRIs), serotonin–norepinephrine reuptake inhibitors (SNRIs), monoamine oxidase inhibitors (MAOIs), and serotonin precursors
5-HT2A_receptor
Abandoned experimental antidepressant drug
the SSRITooltip selective serotonin reuptake inhibitor market in the United States". Serotonin antagonist and reuptake inhibitor List of investigational
Lubazodone
Pharmaceutical compound
also known as midomafetamine or "ecstasy") and the selective serotonin reuptake inhibitor (SSRI) citalopram which is under development for the treatment
MDMA/citalopram
Pharmaceutical compound
the serotonin 5-HT1A, 5-HT2A, 5-HT2B, and 5-HT2C receptors. It is inactive as a serotonin releasing agent and is very weak as a serotonin reuptake inhibitor
5-MeO-NiPT
SSRI drug and metabolite of fluoxetine
Seproxetine, also known as (S)-norfluoxetine, is a selective serotonin reuptake inhibitor (SSRI). It is the (S) enantiomer of norfluoxetine, the active
Seproxetine
Chemical compound
SB-649915 is a serotonin reuptake inhibitor and serotonin 5-HT1A and 5-HT1B receptor antagonist which is being investigated for its antidepressant effects
SB-649915
Selective serotonin reuptake inhibitors, or serotonin-specific re-uptake inhibitor (SSRIs), are a class of chemical compounds that have application as
Development and discovery of SSRI drugs
Development_and_discovery_of_SSRI_drugs
Drug that blocks hallucinogen effects
Examples include serotonin 5-HT1A receptor agonists like buspirone, serotonin reuptake inhibitors such as selective serotonin reuptake inhibitors (SSRIs) like
Trip_killer
Pharmaceutical compound
of the norepinephrine–dopamine reuptake inhibitor (NDRI) bupropion and the serotonin antagonist and reuptake inhibitor (SARI) trazodone which is under
Bupropion/trazodone
Drug class
and 5-hydroxytryptophan (5-HTP), serotonin reuptake inhibitors (SRIs) like selective serotonin reuptake inhibitors (SSRIs) and various other antidepressants
Serotonin 5-HT2A receptor agonist
Serotonin_5-HT2A_receptor_agonist
Pharmaceutical compound
serotonin 5-HT1A receptor. It is also a serotonin reuptake inhibitor, but does not inhibit dopamine or norepinephrine reuptake. The drug shows rather low potency
IPALT
Reversible monoamine oxidase B inhibitor
inhibitors or with drugs that are known to interact with MAO inhibitors, such as pethidine, dextromethorphan, selective serotonin reuptake inhibitors
Safinamide
Investigational narcolepsy and hypersomnia drugs
atypical dopamine reuptake inhibitor (DRI) – idiopathic hypersomnia [32] Golexanolone (GR-3027) – GABAA receptor negative allosteric modulator and neurosteroid
List of investigational narcolepsy and hypersomnia drugs
List_of_investigational_narcolepsy_and_hypersomnia_drugs
NMDA receptor antagonist. It shows a profile of a serotonin–norepinephrine–dopamine reuptake inhibitor (SNDRI). Although this was inferred to be related
PCP_site_2
Class of medications
selective serotonin reuptake inhibitors (SSRIs), serotonin–norepinephrine reuptake inhibitors (SNRIs) and norepinephrine reuptake inhibitors (NRIs). The
Tricyclic_antidepressant
Chemical compound
the serotonin 5-HT7 receptor (ImaxTooltip maximal inhibition = 14%). It is a weak to very weak monoamine reuptake inhibitor, including of serotonin, norepinephrine
Ibogaminalog
Pharmaceutical compound
aorta, which expresses serotonin 5-HT2 receptors. The drug is known to act as a serotonin–norepinephrine–dopamine reuptake inhibitor (SNDRI), with greater
7-Hydroxytryptamine
Pharmaceutical compound
a serotonin 5-HT2A receptor agonist than the known psychedelic drug 5-MeO-iPALT (ASR-3001). The drug is inactive as a monoamine reuptake inhibitor. The
2-Methyl-iPALT
Selective serotonin reuptake inhibitors (SSRIs) (e.g., escitalopram, fluoxetine, paroxetine, sertraline) Serotonin–norepinephrine reuptake inhibitors (SNRIs)
List of psychiatric drugs by type
List_of_psychiatric_drugs_by_type
Metabolite of bupropion
Bupropion is a norepinephrine–dopamine reuptake inhibitor and nicotinic acetylcholine receptor negative allosteric modulator, with its metabolites contributing
Threohydrobupropion
Drug class
that selectively inhibits the action of GABA reuptake and its mechanism of action is the same as selective serotonin reuptake inhibitor (SSRI). It is used
GABA_reuptake_inhibitor
Atypical antidepressant
bupropion, selective serotonin reuptake inhibitors, serotonin-norepinephrine reuptake inhibitors, Monoamine oxidase inhibitor among others) it may also
Tianeptine
Investigational panic disorder drugs
selective serotonin reuptake inhibitor (SSRI) [14] Fluoxetine (LY-110140; Prozac; Reneuron; Sarafem) – selective serotonin reuptake inhibitor (SSRI) [15]
List of investigational panic disorder drugs
List_of_investigational_panic_disorder_drugs
Chemical compound
S33005 is a serotonin–norepinephrine reuptake inhibitor (SNRI) that was under development by Servier for the treatment of depression and related disorders
S33005
Neurotransmission-modulating substance
A serotonin antagonist, or serotonin receptor antagonist, is a drug used to inhibit the action of serotonin and serotonergic drugs at serotonin (5-HT)
Serotonin_receptor_antagonist
Pharmaceutical compound
which acts at multiple targets, being a potent and selective serotonin reuptake inhibitor (SSRI), an agonist of the α2A adrenergic receptor, and a 5-HT2A
Z8779877149
Investigational sexual dysfunction drugs
antidepressant (TCA), serotonin–norepinephrine reuptake inhibitor (SNRI), other actions) and sildenafil (phosphodiesterase PDE5 inhibitor) – premature ejaculation
List of investigational sexual dysfunction drugs
List_of_investigational_sexual_dysfunction_drugs
Chemical compound
TCA. It was thought that TCAs work by inhibiting the reuptake of the neurotransmitters norepinephrine and serotonin by neurons. However, this response occurs
Protriptyline
Chemical compound
humans. 4-MeO-DiPT acts as a serotonin reuptake inhibitor and non-selective serotonin receptor agonist, including of the serotonin 5-HT2A, and 5-HT2C receptors
4-MeO-DiPT
Psychedelic drug
as a serotonin reuptake inhibitor, with low affinity but moderate potency. It shows no activity as a norepinephrine or dopamine reuptake inhibitor. DET
Diethyltryptamine
Chemical compound
tree. It has demonstrated activity as a dopamine reuptake inhibitor, and is also a negative allosteric modulator of the benzodiazepine site of the GABAA
Oroxylin_A
Pharmaceutical compound
acts as a selective atypical serotonin reuptake inhibitor. Specifically, it binds to an allosteric site on the serotonin transporter (SERT), rather than
SNTX-2643
Medication used to treat dyskinesia
doses. It has been found to inhibit the reuptake of serotonin, norepinephrine, and dopamine and to induce the release of serotonin, norepinephrine, and dopamine
Amantadine
Pharmaceutical compound
The drug shows affinity for the serotonin transporter (SERT) (Ki = 172–572 nM). It is a serotonin reuptake inhibitor, with an IC50 value of 1,100 nM.
Pinoline
Opioid analgesic drug
(NOP), as well as an NMDA receptor antagonist and a serotonin-norepinephrine reuptake inhibitor (SNRI). Levorphanol, similarly to certain other opioids
Levorphanol
Atypical antidepressant drug
described as a serotonin antagonist and reuptake inhibitor (SARI) due to its combined actions as a potent antagonist of the serotonin 5-HT2A and 5-HT2C
Nefazodone
Investigational insomnia drugs
(GAT-1) blocker and GABA reuptake inhibitor Triazolam intranasal (Hypnostat; TGAR01H) – GABAA receptor positive allosteric modulator and benzodiazepine
List of investigational insomnia drugs
List_of_investigational_insomnia_drugs
Proteins that function as integral plasma-membrane transporters
classes are serotonin transporters (SERTs), dopamine transporters (DATs), and norepinephrine transporters (NETs) and are responsible for the reuptake of their
Monoamine_transporter
SNRI antidepressant
and has similar effects and pharmacology, acting as a serotonin–norepinephrine reuptake inhibitor. Levomilnacipran was approved for medical use in the
Levomilnacipran
List of pharmaceutical drugs under clinical development for treatment of depression
receptor agonist, serotonin reuptake inhibitor, ionotropic glutamate NMDA receptor antagonist, other actions, and CYP2D6 inhibitor combination Dimethyltryptamine
List of investigational antidepressants
List_of_investigational_antidepressants
Discontinued SSRI antidepressant drug
Indalpine, sold under the brand name Upstène, is a selective serotonin reuptake inhibitor (SSRI) that was briefly marketed as an antidepressant for treatment
Indalpine
Tricyclic antidepressant
et al. (August 1996). "Interactions of selective serotonin reuptake inhibitors with the serotonin 5-HT2c receptor". Psychopharmacology. 126 (3): 234–240
Amitriptyline
travel, tourism, insurance
ALLOSTERIC SEROTONIN-REUPTAKE-INHIBITOR
ALLOSTERIC SEROTONIN-REUPTAKE-INHIBITOR
ALLOSTERIC SEROTONIN-REUPTAKE-INHIBITOR
ALLOSTERIC SEROTONIN-REUPTAKE-INHIBITOR
ALLOSTERIC SEROTONIN-REUPTAKE-INHIBITOR
ALLOSTERIC SEROTONIN-REUPTAKE-INHIBITOR
ALLOSTERIC SEROTONIN-REUPTAKE-INHIBITOR
ALLOSTERIC SEROTONIN-REUPTAKE-INHIBITOR
ALLOSTERIC SEROTONIN-REUPTAKE-INHIBITOR
travel, tourism, insurance